Activity of M3814, an Oral DNA-PK Inhibitor, In Combination with Topoisomerase II Inhibitors in Ovarian Cancer Models. [electronic resource]
- Scientific reports 12 2019
- 18882 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
2045-2322
10.1038/s41598-019-54796-6 doi
Animals Antineoplastic Agents--pharmacology Carcinoma, Ovarian Epithelial--drug therapy Cell Line, Tumor Cell Proliferation--drug effects DNA Damage--drug effects DNA-Activated Protein Kinase--antagonists & inhibitors Doxorubicin--analogs & derivatives Drug Therapy, Combination Etoposide--pharmacology Female Humans Mice Mice, Nude Ovarian Neoplasms--drug therapy Polyethylene Glycols--pharmacology Protein Kinase Inhibitors--pharmacology Topoisomerase II Inhibitors--pharmacology Tumor Burden--drug effects Xenograft Model Antitumor Assays