Badman, Michael K Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of the Novel Non-Bile Acid FXR Agonist Tropifexor (LJN452) in Healthy Volunteers. [electronic resource] - Clinical pharmacology in drug development 04 2020 - 395-410 p. digital Publication Type: Journal Article; Randomized Controlled Trial; Research Support, Non-U.S. Gov't ISSN: 2160-7648 Standard No.: 10.1002/cpdd.762 doi Subjects--Topical Terms: Administration, OralAdultBenzothiazoles--administration & dosageDiet, High-FatDose-Response Relationship, DrugDouble-Blind MethodFastingFemaleFood-Drug InteractionsHalf-LifeHumansIsoxazoles--administration & dosageLipids--bloodMaleMiddle AgedReceptors, Cytoplasmic and Nuclear--agonistsYoung Adult