Corral, Pedro A

Design, synthesis, and enzymatic characterization of quinazoline-based CYP1A2 inhibitors. [electronic resource] - Bioorganic & medicinal chemistry letters 01 2020 - 126719 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1464-3405

10.1016/j.bmcl.2019.126719 doi


Binding Sites
Cytochrome P-450 CYP1A2--chemistry
Cytochrome P-450 CYP1A2 Inhibitors--chemical synthesis
Drug Design
Humans
Molecular Docking Simulation
Protein Structure, Tertiary
Quinazolines--chemistry
Structure-Activity Relationship