Corral, Pedro A
Design, synthesis, and enzymatic characterization of quinazoline-based CYP1A2 inhibitors. [electronic resource]
- Bioorganic & medicinal chemistry letters 01 2020
- 126719 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3405
10.1016/j.bmcl.2019.126719 doi
Binding Sites
Cytochrome P-450 CYP1A2--chemistry
Cytochrome P-450 CYP1A2 Inhibitors--chemical synthesis
Drug Design
Humans
Molecular Docking Simulation
Protein Structure, Tertiary
Quinazolines--chemistry
Structure-Activity Relationship