Pierce, Marquicia R

Syrbactin proteasome inhibitor TIR-199 overcomes bortezomib chemoresistance and inhibits multiple myeloma tumor growth in vivo. [electronic resource] - Leukemia research 01 2020 - 106271 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1873-5835

10.1016/j.leukres.2019.106271 doi


Amides--administration & dosage
Animals
Antineoplastic Combined Chemotherapy Protocols--therapeutic use
Azoles--administration & dosage
Bortezomib--administration & dosage
Cell Line, Tumor
Cell Proliferation--drug effects
Drug Resistance, Neoplasm--drug effects
Drug Synergism
Humans
Male
Mice
Mice, Inbred C57BL
Mice, Inbred NOD
Mice, SCID
Mice, Transgenic
Multiple Myeloma--drug therapy
Peptides, Cyclic--chemistry
Proteasome Inhibitors--administration & dosage
Tumor Burden--drug effects
Xenograft Model Antitumor Assays