Andavar, Sasikumar

Design, Synthesis and Evaluation of Novel Substituted (5-methyl-1H-pyrazol-3-yl)- 1,3,4-oxadiazole as Potent Androgen Receptor Antagonist. [electronic resource] - Anti-cancer agents in medicinal chemistry 2020 - 84-93 p. digital

Publication Type: Journal Article

1875-5992

10.2174/1871520619666191121095720 doi


Androgen Receptor Antagonists--chemical synthesis
Antineoplastic Agents--chemical synthesis
Cell Line, Tumor
Cell Proliferation--drug effects
Cell Survival--drug effects
Dose-Response Relationship, Drug
Drug Design
Drug Screening Assays, Antitumor
Humans
Molecular Docking Simulation
Molecular Structure
Oxadiazoles--chemical synthesis
PC-3 Cells
Receptors, Androgen--genetics
Structure-Activity Relationship