Dopart, Rachel

Allosteric modulators restore orthosteric agonist binding to mutated CB [electronic resource] - The Journal of pharmacy and pharmacology Jan 2020 - 84-91 p. digital

Publication Type: Journal Article

2042-7158

10.1111/jphp.13193 doi


Binding Sites
Cannabinoid Receptor Agonists--metabolism
Cyclohexanols--metabolism
HEK293 Cells
Humans
Indoles--metabolism
Ligands
Mutation
Phenylurea Compounds--metabolism
Piperidines--metabolism
Protein Binding
Protein Conformation
Pyridines--metabolism
Receptor, Cannabinoid, CB1--agonists
Rimonabant--metabolism
Structure-Activity Relationship