Dopart, Rachel Allosteric modulators restore orthosteric agonist binding to mutated CB [electronic resource] - The Journal of pharmacy and pharmacology Jan 2020 - 84-91 p. digital Publication Type: Journal Article ISSN: 2042-7158 Standard No.: 10.1111/jphp.13193 doi Subjects--Topical Terms: Binding SitesCannabinoid Receptor Agonists--metabolismCyclohexanols--metabolismHEK293 CellsHumansIndoles--metabolismLigandsMutationPhenylurea Compounds--metabolismPiperidines--metabolismProtein BindingProtein ConformationPyridines--metabolismReceptor, Cannabinoid, CB1--agonistsRimonabant--metabolismStructure-Activity Relationship