Vergani, Barbara

Novel Benzohydroxamate-Based Potent and Selective Histone Deacetylase 6 (HDAC6) Inhibitors Bearing a Pentaheterocyclic Scaffold: Design, Synthesis, and Biological Evaluation. [electronic resource] - Journal of medicinal chemistry 12 2019 - 10711-10739 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1520-4804

10.1021/acs.jmedchem.9b01194 doi


Animals
Cell Survival--drug effects
Drug Design
Gene Expression Regulation, Enzymologic--drug effects
Histone Deacetylase 6--antagonists & inhibitors
Histones--metabolism
Hydroxamic Acids--chemistry
Mice
Protein Isoforms
Spleen--cytology
T-Lymphocytes, Regulatory
Tubulin--genetics