Vergani, Barbara
Novel Benzohydroxamate-Based Potent and Selective Histone Deacetylase 6 (HDAC6) Inhibitors Bearing a Pentaheterocyclic Scaffold: Design, Synthesis, and Biological Evaluation. [electronic resource]
- Journal of medicinal chemistry 12 2019
- 10711-10739 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1520-4804
10.1021/acs.jmedchem.9b01194 doi
Animals
Cell Survival--drug effects
Drug Design
Gene Expression Regulation, Enzymologic--drug effects
Histone Deacetylase 6--antagonists & inhibitors
Histones--metabolism
Hydroxamic Acids--chemistry
Mice
Protein Isoforms
Spleen--cytology
T-Lymphocytes, Regulatory
Tubulin--genetics