Ebenezer, Oluwakemi

New library of pyrazole-imidazo[1,2-α]pyridine molecular conjugates: Synthesis, antibacterial activity and molecular docking studies. [electronic resource] - Chemical biology & drug design 01 2020 - 162-173 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1747-0285

10.1111/cbdd.13632 doi


Anti-Bacterial Agents--chemical synthesis
Binding Sites
Ciprofloxacin--pharmacology
Drug Evaluation, Preclinical
Drug Resistance, Multiple, Bacterial
Enzyme Inhibitors--chemistry
Glutamine-Fructose-6-Phosphate Transaminase (Isomerizing)--antagonists & inhibitors
Humans
Microbial Sensitivity Tests
Molecular Docking Simulation
Molecular Structure
Pyrazoles--chemical synthesis
Pyridines--chemical synthesis
Small Molecule Libraries--chemical synthesis
Structure-Activity Relationship