In Vitro-In Vivo Inaccuracy: The CYP3A4 Anomaly. [electronic resource]
- Drug metabolism and disposition: the biological fate of chemicals 12 2019
- 1368-1371 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.
1521-009X
10.1124/dmd.119.088427 doi
Cytochrome P-450 CYP3A--metabolism Hepatocytes--drug effects Humans In Vitro Techniques Kinetics Metabolic Clearance Rate Microsomes, Liver--drug effects Models, Biological Pharmaceutical Preparations--metabolism Predictive Value of Tests Substrate Specificity