Hao, Junliang
Synthesis and Pharmacological Characterization of 2-(2,6-Dichlorophenyl)-1-((1 [electronic resource]
- Journal of medicinal chemistry 10 2019
- 8711-8732 p. digital
Publication Type: Journal Article
ISSN: 1520-4804
Standard No.: 10.1021/acs.jmedchem.9b01234 doi
Subjects--Topical Terms: Acetylcholine--metabolism Administration, Oral Allosteric Regulation--drug effects Animals Binding Sites Crystallography, X-Ray Cyclic AMP--metabolism HEK293 Cells Half-Life Humans Isoquinolines--chemistry Kidney--drug effects Locomotion--drug effects Mice Molecular Conformation Protein Isoforms--agonists Rats Receptors, Dopamine D1--agonists Small Molecule Libraries--chemistry Structure-Activity Relationship