Lee, Tobie D

A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. [electronic resource] - Molecular pharmacology 11 2019 - 629-640 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Intramural

1521-0111

10.1124/mol.119.115964 doi


ATP Binding Cassette Transporter, Subfamily B--metabolism
ATP Binding Cassette Transporter, Subfamily B, Member 1--chemistry
ATP Binding Cassette Transporter, Subfamily G, Member 2--metabolism
Antineoplastic Agents--chemistry
Cytotoxins--chemistry
Dose-Response Relationship, Drug
HEK293 Cells
HeLa Cells
High-Throughput Screening Assays--methods
Humans
Neoplasm Proteins--metabolism
Substrate Specificity--drug effects