Cernuda, Bryan

The molecular determinants of R-roscovitine block of hERG channels. [electronic resource] - PloS one 2019 - e0217733 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1932-6203

10.1371/journal.pone.0217733 doi


Animals
Dose-Response Relationship, Drug
Drug Discovery
Ether-A-Go-Go Potassium Channels--antagonists & inhibitors
Humans
Molecular Docking Simulation
Molecular Dynamics Simulation
Molecular Structure
Mutation
Oocytes--drug effects
Potassium Channel Blockers--chemistry
Protein Conformation
Structure-Activity Relationship