Cernuda, Bryan
The molecular determinants of R-roscovitine block of hERG channels. [electronic resource]
- PloS one 2019
- e0217733 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
1932-6203
10.1371/journal.pone.0217733 doi
Animals
Dose-Response Relationship, Drug
Drug Discovery
Ether-A-Go-Go Potassium Channels--antagonists & inhibitors
Humans
Molecular Docking Simulation
Molecular Dynamics Simulation
Molecular Structure
Mutation
Oocytes--drug effects
Potassium Channel Blockers--chemistry
Protein Conformation
Structure-Activity Relationship