TY - GEN AU - Nakagawa,Makoto AU - Nakatani,Fumihiko AU - Matsunaga,Hironori AU - Seki,Takahiko AU - Endo,Makoto AU - Ogawara,Yoko AU - Machida,Yukino AU - Katsumoto,Takuo AU - Yamagata,Kazutsune AU - Hattori,Ayuna AU - Fujita,Shuhei AU - Aikawa,Yukiko AU - Ishikawa,Takamasa AU - Soga,Tomoyoshi AU - Kawai,Akira AU - Chuman,Hirokazu AU - Yokoyama,Nobuhiko AU - Fukushima,Suguru AU - Yahiro,Kenichiro AU - Kimura,Atsushi AU - Shimada,Eijiro AU - Hirose,Takeshi AU - Fujiwara,Toshifumi AU - Setsu,Nokitaka AU - Matsumoto,Yoshihiro AU - Iwamoto,Yukihide AU - Nakashima,Yasuharu AU - Kitabayashi,Issay TI - Selective inhibition of mutant IDH1 by DS-1001b ameliorates aberrant histone modifications and impairs tumor activity in chondrosarcoma SN - 1476-5594 PY - 2020///0226 KW - Bone Neoplasms KW - metabolism KW - Cell Cycle Checkpoints KW - Cell Differentiation KW - Cell Proliferation KW - Chondrosarcoma KW - Enzyme Inhibitors KW - pharmacology KW - Glutarates KW - Histone Code KW - Humans KW - Isocitrate Dehydrogenase KW - antagonists & inhibitors KW - Mutation KW - SOX9 Transcription Factor N1 - Publication Type: Journal Article; Research Support, Non-U.S. Gov't UR - https://doi.org/10.1038/s41388-019-0929-9 ER -