Small molecular modulators of JMJD1C preferentially inhibit growth of leukemia cells. [electronic resource]
- International journal of cancer 01 2020
- 400-412 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1097-0215
10.1002/ijc.32552 doi
Adult Aged Antineoplastic Agents--chemistry Apoptosis--drug effects Bone Marrow--pathology Cell Line, Tumor Cell Proliferation--drug effects DNA Demethylation--drug effects DNA Methylation--drug effects Drug Screening Assays, Antitumor Drug Synergism Female Histones--metabolism Humans Jumonji Domain-Containing Histone Demethylases--antagonists & inhibitors Leukemia, Biphenotypic, Acute--drug therapy Male Middle Aged Molecular Docking Simulation Oxidoreductases, N-Demethylating--antagonists & inhibitors Protein Domains Structure-Activity Relationship Surface Plasmon Resonance Tretinoin--pharmacology