Minh, Nguyen V

Design, Synthesis and Biological Evaluation of Novel N-hydroxyheptanamides Incorporating 6-hydroxy-2-methylquinazolin-4(3H)-ones as Histone Deacetylase Inhibitors and Cytotoxic Agents. [electronic resource] - Anti-cancer agents in medicinal chemistry 2019 - 1543-1557 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1875-5992

10.2174/1871520619666190702142654 doi


Antineoplastic Agents--chemical synthesis
Cell Line, Tumor
Cell Proliferation--drug effects
Dose-Response Relationship, Drug
Drug Design
Drug Screening Assays, Antitumor
Hep G2 Cells
Histone Deacetylase 2--antagonists & inhibitors
Histone Deacetylase Inhibitors--chemical synthesis
Humans
MCF-7 Cells
Molecular Docking Simulation
Molecular Structure
Quinazolines--chemistry
Structure-Activity Relationship