Serafini, Marta

Synthesis, Docking and Biological Evaluation of a Novel Class of Imidazothiazoles as IDO1 Inhibitors. [electronic resource] - Molecules (Basel, Switzerland) May 2019

Publication Type: Journal Article

1420-3049

10.3390/molecules24101874 doi


Binding Sites
Catalytic Domain
Click Chemistry
Enzyme Inhibitors--chemical synthesis
Humans
Imidazoles--chemical synthesis
Indoleamine-Pyrrole 2,3,-Dioxygenase--antagonists & inhibitors
Molecular Conformation
Molecular Docking Simulation
Molecular Dynamics Simulation
Molecular Structure
Protein Binding
Structure-Activity Relationship
Thiazoles--chemical synthesis