Hofman, Jakub

Interactions of Alectinib with Human ATP-Binding Cassette Drug Efflux Transporters and Cytochrome P450 Biotransformation Enzymes: Effect on Pharmacokinetic Multidrug Resistance. [electronic resource] - Drug metabolism and disposition: the biological fate of chemicals 07 2019 - 699-709 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1521-009X

10.1124/dmd.119.086975 doi


ATP-Binding Cassette Transporters--drug effects
Animals
Biotransformation
Carbazoles--pharmacokinetics
Cytochrome P-450 Enzyme System--metabolism
Dogs
Drug Resistance, Multiple--drug effects
Drug Resistance, Neoplasm--drug effects
Humans
Madin Darby Canine Kidney Cells
Piperidines--pharmacokinetics
Protein Kinase Inhibitors--pharmacokinetics