Estimation of competitive antagonist affinity by the Schild method and from functional inhibition curves using a novel form of the Gaddum equation. [electronic resource]
- Toxicology 05 2019
- 21-28 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
1879-3185
10.1016/j.tox.2019.03.015 doi
Animals Benzhydryl Compounds--metabolism Binding, Competitive Dose-Response Relationship, Drug Drug Partial Agonism Endocrine Disruptors--metabolism Estradiol--metabolism Estrogen Receptor Antagonists--metabolism Estrogen Receptor alpha--antagonists & inhibitors Estrogens--metabolism Humans Ligands Models, Biological Phenols--metabolism Protein Binding Reproducibility of Results