Beuckmann, Carsten Theodor Preclinical in vivo characterization of lemborexant (E2006), a novel dual orexin receptor antagonist for sleep/wake regulation. [electronic resource] - Sleep 06 2019 Publication Type: Journal Article; Research Support, Non-U.S. Gov't ISSN: 1550-9109 Standard No.: 10.1093/sleep/zsz076 doi Subjects--Topical Terms: Acetamides--pharmacologyAdrenocorticotropic Hormone--bloodAnimalsFemaleHypnotics and Sedatives--pharmacologyIsoquinolines--pharmacologyMaleMiceMice, Inbred C57BLOrexin Receptor Antagonists--pharmacologyOrexin Receptors--metabolismPyridines--pharmacologyPyrimidines--pharmacologyRatsRats, Sprague-DawleySleep Initiation and Maintenance Disorders--drug therapySleep, REM--drug effectsWakefulness--physiologyZolpidem--pharmacology