Epigenetic Co-Deregulation of EZH2/TET1 is a Senescence-Countering, Actionable Vulnerability in Triple-Negative Breast Cancer. [electronic resource]
- Theranostics 2019
- 761-777 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1838-7640
10.7150/thno.29520 doi
Animals Antibiotics, Antineoplastic--administration & dosage Apoptosis--drug effects Cancer Survivors Cell Line, Tumor Cellular Senescence--drug effects DNA Methylation DNA, Neoplasm--metabolism Doxorubicin--administration & dosage Drug Delivery Systems Enhancer of Zeste Homolog 2 Protein--antagonists & inhibitors Epigenesis, Genetic Female Gene Expression Regulation, Neoplastic--drug effects Humans Indazoles--pharmacology Mice Mice, Nude Mixed Function Oxygenases--antagonists & inhibitors Proto-Oncogene Proteins--antagonists & inhibitors Pyridones--pharmacology Triple Negative Breast Neoplasms--genetics Xenograft Model Antitumor Assays