PROTAC-Mediated Degradation of Bruton's Tyrosine Kinase Is Inhibited by Covalent Binding. [electronic resource]
- ACS chemical biology 03 2019
- 342-347 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1554-8937
10.1021/acschembio.8b01094 doi
Adenine--analogs & derivatives Agammaglobulinaemia Tyrosine Kinase--metabolism Inhibitor of Apoptosis Proteins--metabolism Piperidines Protein Binding Protein Kinase Inhibitors--chemistry Proteolysis Pyrazoles--chemistry Pyrimidines--chemistry Ubiquitin-Protein Ligases--metabolism