Discovery of novel triazolo[4,3-b]pyridazin-3-yl-quinoline derivatives as PIM inhibitors. [electronic resource]
- European journal of medicinal chemistry Apr 2019
- 87-109 p. digital
Publication Type: Journal Article
1768-3254
10.1016/j.ejmech.2019.02.022 doi
Antineoplastic Agents--chemical synthesis Cell Line, Tumor Cell Proliferation--drug effects Dose-Response Relationship, Drug Drug Discovery Drug Screening Assays, Antitumor Humans Molecular Structure Protein Kinase Inhibitors--chemical synthesis Proto-Oncogene Proteins c-pim-1--antagonists & inhibitors Pyridazines--chemical synthesis Quinolines--chemical synthesis Structure-Activity Relationship Triazoles--chemical synthesis