Martínez-González, Sonia

Discovery of novel triazolo[4,3-b]pyridazin-3-yl-quinoline derivatives as PIM inhibitors. [electronic resource] - European journal of medicinal chemistry Apr 2019 - 87-109 p. digital

Publication Type: Journal Article

1768-3254

10.1016/j.ejmech.2019.02.022 doi


Antineoplastic Agents--chemical synthesis
Cell Line, Tumor
Cell Proliferation--drug effects
Dose-Response Relationship, Drug
Drug Discovery
Drug Screening Assays, Antitumor
Humans
Molecular Structure
Protein Kinase Inhibitors--chemical synthesis
Proto-Oncogene Proteins c-pim-1--antagonists & inhibitors
Pyridazines--chemical synthesis
Quinolines--chemical synthesis
Structure-Activity Relationship
Triazoles--chemical synthesis