Complementary activity of tyrosine kinase inhibitors against secondary kit mutations in imatinib-resistant gastrointestinal stromal tumours. [electronic resource]
- British journal of cancer 03 2019
- 612-620 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.
1532-1827
10.1038/s41416-019-0389-6 doi
Animals CHO Cells Clinical Trials, Phase II as Topic Cricetulus Drug Resistance, Neoplasm Female Gastrointestinal Neoplasms--drug therapy Gastrointestinal Stromal Tumors--drug therapy Humans Imatinib Mesylate--pharmacology Mice Mice, Nude Mutation Phenylurea Compounds--pharmacology Protein Kinase Inhibitors--pharmacology Proto-Oncogene Proteins c-kit--antagonists & inhibitors Pyridines--pharmacology Sunitinib--pharmacology Xenograft Model Antitumor Assays