Serrano, César

Complementary activity of tyrosine kinase inhibitors against secondary kit mutations in imatinib-resistant gastrointestinal stromal tumours. [electronic resource] - British journal of cancer 03 2019 - 612-620 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.

1532-1827

10.1038/s41416-019-0389-6 doi


Animals
CHO Cells
Clinical Trials, Phase II as Topic
Cricetulus
Drug Resistance, Neoplasm
Female
Gastrointestinal Neoplasms--drug therapy
Gastrointestinal Stromal Tumors--drug therapy
Humans
Imatinib Mesylate--pharmacology
Mice
Mice, Nude
Mutation
Phenylurea Compounds--pharmacology
Protein Kinase Inhibitors--pharmacology
Proto-Oncogene Proteins c-kit--antagonists & inhibitors
Pyridines--pharmacology
Sunitinib--pharmacology
Xenograft Model Antitumor Assays