Wolle, Patrik

Targeting the MKK7-JNK (Mitogen-Activated Protein Kinase Kinase 7-c-Jun N-Terminal Kinase) Pathway with Covalent Inhibitors. [electronic resource] - Journal of medicinal chemistry 03 2019 - 2843-2848 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1520-4804

10.1021/acs.jmedchem.9b00102 doi


Crystallography, X-Ray
Drug Design
JNK Mitogen-Activated Protein Kinases--antagonists & inhibitors
MAP Kinase Kinase 7--antagonists & inhibitors
Phosphorylation
Protein Kinase Inhibitors--chemistry
Pyrazoles--chemistry
Pyrimidines--chemistry