Stanczyk, M Alexander

The δ-opioid receptor positive allosteric modulator BMS 986187 is a G-protein-biased allosteric agonist. [electronic resource] - British journal of pharmacology 06 2019 - 1649-1663 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1476-5381

10.1111/bph.14602 doi


Allosteric Site
Animals
CHO Cells
Cricetulus
GTP-Binding Proteins--agonists
Guanosine 5'-O-(3-Thiotriphosphate)--metabolism
HEK293 Cells
Humans
Male
Mice
Receptors, Opioid, delta--metabolism
Xanthones--pharmacology