The δ-opioid receptor positive allosteric modulator BMS 986187 is a G-protein-biased allosteric agonist. [electronic resource]
- British journal of pharmacology 06 2019
- 1649-1663 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
1476-5381
10.1111/bph.14602 doi
Allosteric Site Animals CHO Cells Cricetulus GTP-Binding Proteins--agonists Guanosine 5'-O-(3-Thiotriphosphate)--metabolism HEK293 Cells Humans Male Mice Receptors, Opioid, delta--metabolism Xanthones--pharmacology