TY  - GEN
AU  - Kalyukina,Maria
AU  - Yosaatmadja,Yuliana
AU  - Middleditch,Martin J
AU  - Patterson,Adam V
AU  - Smaill,Jeff B
AU  - Squire,Christopher J
TI  - TAS-120 Cancer Target Binding: Defining Reactivity and Revealing the First Fibroblast Growth Factor Receptor 1 (FGFR1) Irreversible Structure
SN  - 1860-7187
PY  - 2019///1125
KW  - Binding Sites
KW  - Cell Line, Tumor
KW  - Crystallography, X-Ray
KW  - Humans
KW  - Molecular Dynamics Simulation
KW  - Protein Structure, Tertiary
KW  - Pyrazoles
KW  - chemistry
KW  - Pyrimidines
KW  - Receptor, Fibroblast Growth Factor, Type 1
KW  - antagonists & inhibitors
KW  - Recombinant Proteins
KW  - biosynthesis
N1  - Publication Type: Journal Article; Research Support, Non-U.S. Gov't
UR  - https://doi.org/10.1002/cmdc.201800719
ER  -