Kalyukina, Maria

TAS-120 Cancer Target Binding: Defining Reactivity and Revealing the First Fibroblast Growth Factor Receptor 1 (FGFR1) Irreversible Structure. [electronic resource] - ChemMedChem 02 2019 - 494-500 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1860-7187

10.1002/cmdc.201800719 doi


Binding Sites
Cell Line, Tumor
Crystallography, X-Ray
Humans
Molecular Dynamics Simulation
Protein Structure, Tertiary
Pyrazoles--chemistry
Pyrimidines--chemistry
Receptor, Fibroblast Growth Factor, Type 1--antagonists & inhibitors
Recombinant Proteins--biosynthesis