Barinka, Cyril

Structural and computational basis for potent inhibition of glutamate carboxypeptidase II by carbamate-based inhibitors. [electronic resource] - Bioorganic & medicinal chemistry 01 2019 - 255-264 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't

1464-3391

10.1016/j.bmc.2018.11.022 doi


Animals
Carbamates--chemical synthesis
Catalytic Domain
Cell Line
Drosophila--genetics
Enzyme Assays
Glutamate Carboxypeptidase II--antagonists & inhibitors
Humans
Hydrogen Bonding
Models, Molecular
Protease Inhibitors--chemical synthesis
Protein Binding
Quantum Theory
Stereoisomerism
Urea--analogs & derivatives