Fluorine-18 isotope labeling for positron emission tomography imaging. Direct evidence for DBPR211 as a peripherally restricted CB1 inverse agonist. [electronic resource]
- Bioorganic & medicinal chemistry 01 2019
- 216-223 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3391
10.1016/j.bmc.2018.11.043 doi
Animals Cannabinoid Receptor Agonists--chemical synthesis Drug Inverse Agonism Fluorine Radioisotopes Isotope Labeling Male Mice, Inbred C57BL Positron-Emission Tomography--methods Pyrazoles--chemical synthesis Receptor, Cannabinoid, CB1--agonists Sulfonamides--chemical synthesis Thiophenes--chemistry Tissue Distribution