Metabolic targeting synergizes with MAPK inhibition and delays drug resistance in melanoma. [electronic resource]
- Cancer letters 02 2019
- 453-463 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1872-7980
10.1016/j.canlet.2018.11.018 doi
Anti-Inflammatory Agents, Non-Steroidal--pharmacology Antineoplastic Combined Chemotherapy Protocols--pharmacology Apoptosis--drug effects Cell Line, Tumor Cell Proliferation--drug effects Diclofenac--analogs & derivatives Dose-Response Relationship, Drug Drug Resistance, Neoplasm--drug effects Drug Synergism Energy Metabolism--drug effects Genetic Predisposition to Disease Humans Melanoma--drug therapy Mitogen-Activated Protein Kinases--antagonists & inhibitors Mutation Phenotype Protein Kinase Inhibitors--pharmacology Proto-Oncogene Proteins B-raf--antagonists & inhibitors Signal Transduction--drug effects Skin Neoplasms--drug therapy Time Factors Vemurafenib--pharmacology