Pereira, Adriana S A

Inhibition of histone methyltransferase EZH2 in Schistosoma mansoni in vitro by GSK343 reduces egg laying and decreases the expression of genes implicated in DNA replication and noncoding RNA metabolism. [electronic resource] - PLoS neglected tropical diseases 10 2018 - e0006873 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1935-2735

10.1371/journal.pntd.0006873 doi


Animals
DNA Replication--drug effects
Enhancer of Zeste Homolog 2 Protein--antagonists & inhibitors
Enzyme Inhibitors--pharmacology
Female
Gene Expression Regulation--drug effects
Indazoles--pharmacology
Locomotion--drug effects
Male
Metabolic Networks and Pathways--drug effects
Microscopy, Electron, Scanning
Oviposition--drug effects
Pyridones--pharmacology
RNA, Untranslated--metabolism
Schistosoma mansoni--drug effects
Survival Analysis