TY  - GEN
AU  - Yang,Shyh-Ming
AU  - Urban,Daniel J
AU  - Yoshioka,Makoto
AU  - Strovel,Jeffrey W
AU  - Fletcher,Steven
AU  - Wang,Amy Q
AU  - Xu,Xin
AU  - Shah,Pranav
AU  - Hu,Xin
AU  - Hall,Matthew D
AU  - Jadhav,Ajit
AU  - Maloney,David J
TI  - Discovery and lead identification of quinazoline-based BRD4 inhibitors
SN  - 1464-3405
PY  - 2019///0514
KW  - Animals
KW  - Binding Sites
KW  - Cell Cycle Proteins
KW  - Cell Line, Tumor
KW  - Drug Discovery
KW  - Humans
KW  - Mice
KW  - Microsomes, Liver
KW  - metabolism
KW  - Molecular Structure
KW  - Nuclear Proteins
KW  - antagonists & inhibitors
KW  - Quinazolines
KW  - chemical synthesis
KW  - Structure-Activity Relationship
KW  - Transcription Factors
N1  - Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, N.I.H., Intramural
UR  - https://doi.org/10.1016/j.bmcl.2018.08.039
ER  -