Strategy for Tumor-Selective Disruption of Androgen Receptor Function in the Spectrum of Prostate Cancer. [electronic resource]
- Clinical cancer research : an official journal of the American Association for Cancer Research 12 2018
- 6509-6522 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, U.S. Gov't, Non-P.H.S.
1557-3265
10.1158/1078-0432.CCR-18-0982 doi
Androgen Receptor Antagonists--chemistry Animals Antineoplastic Agents, Hormonal--chemistry Cell Line, Tumor Disease Models, Animal Drug Discovery--methods Drug Screening Assays, Antitumor Gene Expression Profiling High-Throughput Screening Assays Humans Male Mice Promoter Regions, Genetic Prostatic Neoplasms--drug therapy Protein Binding Receptors, Androgen--metabolism Structure-Activity Relationship Xenograft Model Antitumor Assays ets-Domain Protein Elk-1--metabolism