Piemontese, Luca

Donepezil structure-based hybrids as potential multifunctional anti-Alzheimer's drug candidates. [electronic resource] - Journal of enzyme inhibition and medicinal chemistry Dec 2018 - 1212-1224 p. digital

Publication Type: Journal Article

1475-6374

10.1080/14756366.2018.1491564 doi


Acetylcholinesterase--metabolism
Alzheimer Disease--drug therapy
Amyloid beta-Peptides--antagonists & inhibitors
Antioxidants--chemical synthesis
Caco-2 Cells
Cell Line, Tumor
Cell Survival--drug effects
Cholinesterase Inhibitors--chemical synthesis
Donepezil
Dose-Response Relationship, Drug
Humans
Indans--chemical synthesis
Models, Molecular
Molecular Structure
Piperidines--chemical synthesis
Protein Aggregates--drug effects
Structure-Activity Relationship