Kassab, Asmaa E

Novel benzotriazole N-acylarylhydrazone hybrids: Design, synthesis, anticancer activity, effects on cell cycle profile, caspase-3 mediated apoptosis and FAK inhibition. [electronic resource] - Bioorganic chemistry 10 2018 - 531-544 p. digital

Publication Type: Journal Article

1090-2120

10.1016/j.bioorg.2018.07.008 doi


Antineoplastic Agents--chemical synthesis
Apoptosis--drug effects
Caspase 3--metabolism
Cell Cycle--drug effects
Cell Line, Tumor
Cell Proliferation--drug effects
Drug Design
Drug Screening Assays, Antitumor
Focal Adhesion Protein-Tyrosine Kinases--antagonists & inhibitors
Humans
Hydrazones--chemical synthesis
Molecular Docking Simulation
Neoplasms--drug therapy
Triazoles--chemical synthesis