In vitro and ex vivo anti-fibrotic effects of LY2109761, a small molecule inhibitor against TGF-β. [electronic resource]
- Toxicology and applied pharmacology 09 2018
- 127-137 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1096-0333
10.1016/j.taap.2018.07.001 doi
Adenosine Triphosphate--metabolism Animals Cell Line Collagen Type I--antagonists & inhibitors Down-Regulation Fibrosis--drug therapy Gene Expression--drug effects Humans In Vitro Techniques Liver--drug effects Male Phosphorylation Pyrazoles--pharmacology Pyrroles--pharmacology Rats Rats, Wistar Smad1 Protein--antagonists & inhibitors Smad2 Protein--antagonists & inhibitors Tissue Inhibitor of Metalloproteinase-2--antagonists & inhibitors Transforming Growth Factor beta--antagonists & inhibitors