Single Nucleotide Polymorphisms (SNPs) Distant from Xenobiotic Response Elements Can Modulate Aryl Hydrocarbon Receptor Function: SNP-Dependent CYP1A1 Induction. [electronic resource]
- Drug metabolism and disposition: the biological fate of chemicals 09 2018
- 1372-1381 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural
1521-009X
10.1124/dmd.118.082164 doi
5' Untranslated Regions Basic Helix-Loop-Helix Transcription Factors--agonists Binding Sites Cell Line, Tumor Cytochrome P-450 CYP1A1--biosynthesis Cytochrome P-450 Enzyme Inducers--pharmacology Enzyme Induction Humans Methylcholanthrene--pharmacology Polymorphism, Single Nucleotide Protein Binding Receptors, Aryl Hydrocarbon--agonists Response Elements Transcription, Genetic Xenobiotics--metabolism