Bapiro, Tashinga E <br/><br/>
Complete Substrate Inhibition of Cytochrome P450 2C8 by AZD9496, an Oral Selective Estrogen Receptor Degrader.  [electronic resource] 

 -  Drug metabolism and disposition: the biological fate of chemicals  09 2018 
 - 1268-1276 p.  digital 
<br/><br/> Publication Type: Journal Article; Research Support, Non-U.S. Gov't 
<br/><br/><label>ISSN: </label>1521-009X 
<br/><br/><label>Standard No.: </label>10.1124/dmd.118.081539  doi 
<br/><br/><label>Subjects--Topical Terms: </label><br/>Administration, Oral<br/>Cinnamates--metabolism<br/>Cytochrome P-450 CYP2C8--metabolism<br/>Cytochrome P-450 CYP2C8 Inhibitors--metabolism<br/>Dose-Response Relationship, Drug<br/>Female<br/>Humans<br/>Indoles--metabolism<br/>Male<br/>Microsomes, Liver--drug effects<br/>Receptors, Estrogen--antagonists & inhibitors<br/>Substrate Specificity--drug effects