TY - GEN AU - Magliocca,Salvatore AU - De Caro,Carmen AU - Lazzarato,Loretta AU - Russo,Roberto AU - Rolando,Barbara AU - Chegaev,Konstantin AU - Marini,Elisabetta AU - Nieddu,Maria AU - Burrai,Lucia AU - Boatto,Gianpiero AU - Cristiano,Claudia AU - Marabello,Domenica AU - Gazzano,Elena AU - Riganti,Chiara AU - Sodano,Federica AU - Rimoli,Maria Grazia TI - Aceclofenac-Galactose Conjugate: Design, Synthesis, Characterization, and Pharmacological and Toxicological Evaluations SN - 1543-8392 PY - 2019///0723 KW - Acute Pain KW - drug therapy KW - Administration, Oral KW - Animals KW - Anti-Inflammatory Agents, Non-Steroidal KW - administration & dosage KW - Biological Availability KW - Caco-2 Cells KW - Carrageenan KW - toxicity KW - Diclofenac KW - Disease Models, Animal KW - Drug Carriers KW - chemistry KW - Drug Compounding KW - methods KW - Edema KW - chemically induced KW - Galactose KW - Gastric Mucosa KW - drug effects KW - Humans KW - Hydrolysis KW - Intestinal Mucosa KW - Male KW - Mice KW - Permeability KW - Platelet Aggregation KW - Prodrugs KW - Solubility KW - Stomach Ulcer N1 - Publication Type: Journal Article UR - https://doi.org/10.1021/acs.molpharmaceut.8b00195 ER -