Magliocca, Salvatore
Aceclofenac-Galactose Conjugate: Design, Synthesis, Characterization, and Pharmacological and Toxicological Evaluations. [electronic resource]
- Molecular pharmaceutics 08 2018
- 3101-3110 p. digital
Publication Type: Journal Article
1543-8392
10.1021/acs.molpharmaceut.8b00195 doi
Acute Pain--drug therapy
Administration, Oral
Animals
Anti-Inflammatory Agents, Non-Steroidal--administration & dosage
Biological Availability
Caco-2 Cells
Carrageenan--toxicity
Diclofenac--administration & dosage
Disease Models, Animal
Drug Carriers--chemistry
Drug Compounding--methods
Edema--chemically induced
Galactose--chemistry
Gastric Mucosa--drug effects
Humans
Hydrolysis
Intestinal Mucosa--drug effects
Male
Mice
Permeability
Platelet Aggregation--drug effects
Prodrugs--administration & dosage
Solubility
Stomach Ulcer--chemically induced