Ling, Yong

Development of novel amino-quinoline-5,8-dione derivatives as NAD(P)H:quinone oxidoreductase 1 (NQO1) inhibitors with potent antiproliferative activities. [electronic resource] - European journal of medicinal chemistry Jun 2018 - 199-209 p. digital

Publication Type: Journal Article

1768-3254

10.1016/j.ejmech.2018.05.025 doi


Antineoplastic Agents--chemical synthesis
Cell Line, Tumor
Cell Proliferation--drug effects
Dose-Response Relationship, Drug
Drug Screening Assays, Antitumor
Enzyme Inhibitors--chemical synthesis
Humans
Molecular Structure
NAD(P)H Dehydrogenase (Quinone)--antagonists & inhibitors
Quinolones--chemical synthesis
Structure-Activity Relationship