Artschwager, Raik

Potent and Highly Selective Inhibitors of the Proteasome Trypsin-like Site by Incorporation of Basic Side Chain Containing Amino Acid Derived Sulfonyl Fluorides. [electronic resource] - Journal of medicinal chemistry 06 2018 - 5395-5411 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1520-4804

10.1021/acs.jmedchem.8b00685 doi


Amino Acids--chemistry
Drug Evaluation, Preclinical--methods
Humans
Proteasome Endopeptidase Complex--chemistry
Proteasome Inhibitors--chemistry
Structure-Activity Relationship
Sulfinic Acids--chemistry
Trypsin--chemistry