Discovery of coumarin-dihydroquinazolinone analogs as niacin receptor 1 agonist with in-vivo anti-obesity efficacy. [electronic resource]
- European journal of medicinal chemistry May 2018
- 208-222 p. digital
Publication Type: Journal Article
1768-3254
10.1016/j.ejmech.2018.04.037 doi
Animals Anti-Obesity Agents--chemical synthesis Coumarins--chemical synthesis Diet, High-Fat--adverse effects Dose-Response Relationship, Drug Drug Discovery Glucose Tolerance Test Male Mice Mice, Inbred C57BL Models, Molecular Molecular Structure Obesity--chemically induced Quinazolinones--chemical synthesis Receptors, G-Protein-Coupled--agonists Receptors, Nicotinic Structure-Activity Relationship