Mitra, Pallabi

Prediction and Quantification of Hepatic Transporter-Mediated Uptake of Pitavastatin Utilizing a Combination of the Relative Activity Factor Approach and Mechanistic Modeling. [electronic resource] - Drug metabolism and disposition: the biological fate of chemicals 07 2018 - 953-963 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1521-009X

10.1124/dmd.118.080614 doi


Adult
Biological Transport--physiology
Cell Line
Cyclosporine--metabolism
Drug Interactions--physiology
Female
HEK293 Cells
Hepatocytes--drug effects
Humans
Hydroxymethylglutaryl-CoA Reductase Inhibitors--metabolism
Liver--drug effects
Liver-Specific Organic Anion Transporter 1--metabolism
Male
Membrane Transport Proteins--metabolism
Middle Aged
Organic Anion Transporters, Sodium-Dependent--metabolism
Quinolines--metabolism
Rifampin--metabolism
Solute Carrier Organic Anion Transporter Family Member 1B3--metabolism
Symporters--metabolism