Agarwal, Sameer

Evaluation of novel TGR5 agonist in combination with Sitagliptin for possible treatment of type 2 diabetes. [electronic resource] - Bioorganic & medicinal chemistry letters 06 2018 - 1849-1852 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1464-3405

10.1016/j.bmcl.2018.04.011 doi


Animals
Binding Sites
Diabetes Mellitus, Type 2--drug therapy
Drug Therapy, Combination
Female
Glucagon-Like Peptide 1--metabolism
Half-Life
Humans
Hypoglycemic Agents--chemistry
Imidazoles--chemistry
Mice
Mice, Inbred C57BL
Molecular Docking Simulation
Protein Structure, Tertiary
Receptors, G-Protein-Coupled--agonists
Sitagliptin Phosphate--therapeutic use
Structure-Activity Relationship