Evaluation of novel TGR5 agonist in combination with Sitagliptin for possible treatment of type 2 diabetes. [electronic resource]
- Bioorganic & medicinal chemistry letters 06 2018
- 1849-1852 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1464-3405
10.1016/j.bmcl.2018.04.011 doi
Animals Binding Sites Diabetes Mellitus, Type 2--drug therapy Drug Therapy, Combination Female Glucagon-Like Peptide 1--metabolism Half-Life Humans Hypoglycemic Agents--chemistry Imidazoles--chemistry Mice Mice, Inbred C57BL Molecular Docking Simulation Protein Structure, Tertiary Receptors, G-Protein-Coupled--agonists Sitagliptin Phosphate--therapeutic use Structure-Activity Relationship