Mou, Jianfeng

Structure-activity relationship study of a series of caspase inhibitors containing γ-amino acid moiety for treatment of cholestatic liver disease. [electronic resource] - Bioorganic & medicinal chemistry letters 06 2018 - 1874-1878 p. digital

Publication Type: Journal Article

1464-3405

10.1016/j.bmcl.2018.04.002 doi


Amino Acids--chemistry
Animals
Bilirubin--blood
Binding Sites
Caspase 1--chemistry
Caspase Inhibitors--chemistry
Disease Models, Animal
Half-Life
Humans
Jurkat Cells
Liver Diseases--drug therapy
Mice
Molecular Docking Simulation
Protein Structure, Tertiary
Structure-Activity Relationship
fas Receptor--antagonists & inhibitors