Ménard, Ludovic
Reactivation of Mutant-EGFR Degradation through Clathrin Inhibition Overcomes Resistance to EGFR Tyrosine Kinase Inhibitors. [electronic resource]
- Cancer research 06 2018
- 3267-3279 p. digital
Publication Type: Journal Article
ISSN: 1538-7445
Standard No.: 10.1158/0008-5472.CAN-17-2195 doi
Subjects--Topical Terms: Antineoplastic Combined Chemotherapy Protocols--pharmacology Apoptosis--drug effects Carcinoma, Non-Small-Cell Lung--drug therapy Cell Line, Tumor Clathrin--antagonists & inhibitors Drug Resistance, Neoplasm--drug effects Endocytosis--drug effects ErbB Receptors--genetics Humans Lung Neoplasms--drug therapy Lysosomes--metabolism Mutation Protein Kinase Inhibitors--pharmacology Proteolysis--drug effects Signal Transduction--genetics Sulfonamides--pharmacology Thiazolidines--pharmacology