TY - GEN AU - Patel,Hetal AU - Periyasamy,Manikandan AU - Sava,Georgina P AU - Bondke,Alexander AU - Slafer,Brian W AU - Kroll,Sebastian H B AU - Barbazanges,Marion AU - Starkey,Richard AU - Ottaviani,Silvia AU - Harrod,Alison AU - Aboagye,Eric O AU - Buluwela,Laki AU - Fuchter,Matthew J AU - Barrett,Anthony G M AU - Coombes,R Charles AU - Ali,Simak TI - ICEC0942, an Orally Bioavailable Selective Inhibitor of CDK7 for Cancer Treatment SN - 1538-8514 PY - 2019///0625 KW - Administration, Oral KW - Animals KW - Antineoplastic Agents KW - administration & dosage KW - Biological Availability KW - Caspases KW - metabolism KW - Cell Cycle KW - drug effects KW - Cell Line, Tumor KW - Cyclin-Dependent Kinases KW - antagonists & inhibitors KW - Disease Models, Animal KW - Dose-Response Relationship, Drug KW - Humans KW - Mice KW - Phosphorylation KW - Protein Kinase Inhibitors KW - Xenograft Model Antitumor Assays KW - Cyclin-Dependent Kinase-Activating Kinase N1 - Publication Type: Journal Article; Research Support, Non-U.S. Gov't UR - https://doi.org/10.1158/1535-7163.MCT-16-0847 ER -