Helliwell, Matthew V

Structural implications of hERG K [electronic resource] - The Journal of biological chemistry 05 2018 - 7040-7057 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1083-351X

10.1074/jbc.RA117.000363 doi


Alanine--chemistry
Computer Simulation
Cryoelectron Microscopy
Crystallography, X-Ray
Dose-Response Relationship, Drug
ERG1 Potassium Channel--antagonists & inhibitors
HEK293 Cells
Humans
Inhibitory Concentration 50
Ion Channel Gating--drug effects
Molecular Docking Simulation
Mutation
Patch-Clamp Techniques
Phenylalanine--chemistry
Potassium Channel Blockers--administration & dosage
Protein Binding
Protein Conformation