Binding Mode Characterization and Early in Vivo Evaluation of Fragment-Like Thiols as Inhibitors of the Virulence Factor LasB from Pseudomonas aeruginosa. [electronic resource]
- ACS infectious diseases 06 2018
- 988-997 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
2373-8227
10.1021/acsinfecdis.8b00010 doi
Animals Anti-Bacterial Agents--chemical synthesis Bacterial Proteins--antagonists & inhibitors Binding Sites Cell Line Chromatography, Liquid Drug Evaluation, Preclinical Drug Resistance, Bacterial Humans Mass Spectrometry Metalloendopeptidases--antagonists & inhibitors Models, Molecular Molecular Conformation Molecular Structure Moths--microbiology Protein Binding Pseudomonas aeruginosa--drug effects Structure-Activity Relationship Sulfhydryl Compounds--chemical synthesis Virulence Factors