Kany, Andreas M

Binding Mode Characterization and Early in Vivo Evaluation of Fragment-Like Thiols as Inhibitors of the Virulence Factor LasB from Pseudomonas aeruginosa. [electronic resource] - ACS infectious diseases 06 2018 - 988-997 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

2373-8227

10.1021/acsinfecdis.8b00010 doi


Animals
Anti-Bacterial Agents--chemical synthesis
Bacterial Proteins--antagonists & inhibitors
Binding Sites
Cell Line
Chromatography, Liquid
Drug Evaluation, Preclinical
Drug Resistance, Bacterial
Humans
Mass Spectrometry
Metalloendopeptidases--antagonists & inhibitors
Models, Molecular
Molecular Conformation
Molecular Structure
Moths--microbiology
Protein Binding
Pseudomonas aeruginosa--drug effects
Structure-Activity Relationship
Sulfhydryl Compounds--chemical synthesis
Virulence Factors